Accepted Name |
17alpha-hydroxyprogesterone deacetylase
|
Alternative Name(s) |
17alpha-hydroxyprogesterone 17,20-lyase |
17alpha-hydroxyprogesterone acetaldehyde-lyase |
CYP17 |
CYP17A1 |
Reaction catalysed |
- 17alpha-hydroxyprogesterone + O2 + reduced [NADPH--hemoprotein reductase] = acetate + androst-4-ene-3,17-dione + 2 H(+) + H2O + oxidized [NADPH--hemoprotein reductase]
- 17alpha-hydroxypregnenolone + O2 + reduced [NADPH--hemoprotein reductase] = 3beta-hydroxyandrost-5-en-17-one + acetate + 2 H(+) + H2O + oxidized [NADPH--hemoprotein reductase]
|
Comment(s) |
- A microsomal protein that catalyzes two independent reactions at the
same active site - the 17-hydroxylation of pregnenolone and
progesterone, which is part of glucocorticoid hormones biosynthesis
(EC 1.14.14.19), and the conversion of the 17-hydroxylated products
via a 17,20-lyase reaction to form androstenedione and 3beta-
hydroxyandrost-5-en-17-one, leading to sex hormone biosynthesis.
- The activity of this reaction is dependent on the allosteric
interaction of the enzyme with cytochrome b5 without any transfer of
electrons from the cytochrome.
- The enzymes from different organisms differ in their substrate
specificity; while the enzymes from pig, hamster, and rat accept both
17alpha-hydroxyprogesterone and 17alpha-hydroxypregnenolone,
the enzymes from human, bovine, sheep, goat, and bison do not accept
the former, and the enzyme from guinea pig does not accept the
latter.
- Formerly EC 4.1.2.30.
|
Cross-references |
BRENDA | 1.14.14.32 |
EC2PDB | 1.14.14.32 |
ExplorEnz | 1.14.14.32 |
PRIAM enzyme-specific profiles | 1.14.14.32 |
KEGG Ligand Database for Enzyme Nomenclature | 1.14.14.32 |
IUBMB Enzyme Nomenclature | 1.14.14.32 |
IntEnz | 1.14.14.32 |
MEDLINE | Find literature relating to 1.14.14.32 |
MetaCyc | 1.14.14.32 |
Rhea expert-curated reactions | 1.14.14.32 |
UniProtKB/Swiss-Prot |
Q9GMC7, CP17A_BISBI | P05185, CP17A_BOVIN | Q9N0U7, CP17A_CAPHI |
Q64410, CP17A_CAVPO | P12394, CP17A_CHICK | Q9GMC8, CP17A_FELCA |
Q95328, CP17A_HORSE | P05093, CP17A_HUMAN | O73853, CP17A_ICTPU |
Q2XVA1, CP17A_MACFA | Q8HYM9, CP17A_MACMU | P70687, CP17A_MESAU |
P27786, CP17A_MOUSE | P30437, CP17A_ONCMY | P70085, CP17A_ORYLA |
Q8HYN1, CP17A_PANTR | Q8HYN0, CP17A_PAPCY | Q9GLD2, CP17A_PAPHU |
Q91Z85, CP17A_PERLE | P19100, CP17A_PIG | O57525, CP17A_RANDY |
P11715, CP17A_RAT | Q29497, CP17A_SHEEP | Q92113, CP17A_SQUAC |
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