ENZYME entry: EC 2.7.11.15
Accepted Name |
[beta-adrenergic-receptor] kinase.
|
Alternative Name(s) |
ADRBK1. |
adrenergic receptor kinase. |
BARK1. |
beta2ARK. |
beta-adrenergic-receptor kinase. |
beta-adrenergic-receptor kinase (phosphorylating). |
beta-adrenergic receptor-specific kinase. |
beta-adrenoceptor kinase. |
beta-ARK. |
beta-AR kinase. |
beta-receptor kinase. |
Reaction catalysed |
[beta-adrenergic receptor] + ATP <=> [beta-adrenergic receptor]-phosphate + ADP + H(+) |
Comment(s) |
- Acts on the agonist-occupied form of the receptor; also
phosphorylates rhodopsin, but more slowly.
- Does not act on casein or histones.
- Inhibited by Zn(2+) and digitonin but is unaffected by cyclic-AMP
(cf. EC 2.7.11.14 and EC 2.7.11.16).
- Formerly EC 2.7.1.126.
|
Cross-references |
BRENDA | 2.7.11.15 |
EC2PDB | 2.7.11.15 |
ExplorEnz | 2.7.11.15 |
PRIAM enzyme-specific profiles | 2.7.11.15 |
KEGG Ligand Database for Enzyme Nomenclature | 2.7.11.15 |
IUBMB Enzyme Nomenclature | 2.7.11.15 |
IntEnz | 2.7.11.15 |
MEDLINE | Find literature relating to 2.7.11.15 |
MetaCyc | 2.7.11.15 |
Rhea expert-curated reactions | 2.7.11.15 |
UniProtKB/Swiss-Prot |
P21146, ARBK1_BOVIN; | O97627, ARBK1_DIDVI; | P25098, ARBK1_HUMAN; |
Q64682, ARBK1_MESAU; | Q99MK8, ARBK1_MOUSE; | P26817, ARBK1_RAT; |
P26818, ARBK2_BOVIN; | P35626, ARBK2_HUMAN; | Q3UYH7, ARBK2_MOUSE; |
P26819, ARBK2_RAT; |
|
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